Chemical Name/IUPAC:(2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-((((1r,3S)-3-(2-(5-(tert-butyl)-1H-benzo[d]imidazol-2-yl)ethyl)cyclobutyl)(isopropyl)amino)methyl)tetrahydrofuran-3,4-diolTechnical Data
Product Name: EPZ-5676 (Pinometostat)
Chemical Formula: C30H42N8O3
Molecular Weight: 562.7
CAS#: 1380288-87-8
Appearance: Solid powder
Purity: > 99% by HPLC
Solubility: Soluble in DMSO
Storage: Room temperature for months, or -20oC for 3 yearsDescription EPZ-5676 (Pinometostat) is a small molecule inhibitor of histone methyltransferase with potential antineoplastic activity. Upon intravenous administration, EPZ-5676 specifically blocks the activity of the histone lysine-methyltransferase DOT1L, thereby inhibiting the methylation of nucleosomal histone H3 on lysine 79 (H3K79) that is bound to the mixed lineage leukemia (MLL) fusion protein which targets genes and blocks the expression of leukemogenic genes.
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Isabella Scott - 2024-03-03
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Isabella Clark - 2024-03-03
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Harper Lee - 2024-03-03
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Isabella Scott - 2024-03-03
Truly a step above the rest in terms of quality and service. The delivery was swift, and the product is worth every penny!